SB-715992

• CAT Number: I003220
• CAS Number: 336113-53-2
• Molecular Formula: C₃₀H₃₃ClN₄O₂
• Molecular Weight: 517.06
• Purity: ≥95%
• Target: Ksp
• Solubility: DMSO 100 mg/mL Ethanol 100 mg/mL
• Storage: 3 years -20C powder
• IC50: 1.7 nM(Ki)
• InChI: InChI=1S/C30H33ClN4O2/c1-20(2)27(34(17-7-16-32)29(36)23-12-10-21(3)11-13-23)28-33-26-18-24(31)14-15-25(26)30(37)35(28)19-22-8-5-4-6-9-22/h4-6,8-15,18,20,27H,7,16-17,19,32H2,1-3H3/t27-/m1/s1
• InChIKey: QJZRFPJCWMNVAV-HHHXNRCGSA-N
• SMILES: CC1=CC=C(C=C1)C(=O)N(CCCN)C(C2=NC3=C(C=CC(=C3)Cl)C(=O)N2CC4=CC=CC=C4)C(C)C

SB-715992 (Cat.No:I003220) is a chemical compound and a potent inhibitor of cyclin-dependent kinases (CDKs). It is being studied for its potential in cancer therapy due to its ability to halt cell cycle progression and induce apoptosis in cancer cells. SB-715992 shows promise as a targeted therapeutic agent for various malignancies.

Reference

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