For research use only. Not for therapeutic Use.
Plecstatin-1 hydrochloride(CAT: I040277) is a unique organoeuropium-based anticancer agent that selectively targets plectin, a cytolinker protein involved in maintaining cellular architecture and signaling. Plectin is often overexpressed or mislocalized in cancer cells, making it an attractive therapeutic target. Plecstatin-1 exhibits selective accumulation in tumor spheroids, where it disrupts cellular structure and impairs tumor viability. Its europium coordination enhances molecular tracking and imaging potential, offering dual functionality for therapy and visualization. This compound is a valuable tool for cancer biology research, particularly in studies of cytoskeletal disruption and targeted cancer therapy.
Molecular Formula | C22H24Cl3FN2RuS |
Purity | ≥95% |
Chemistry Calculators | Dilution Calculator In vivo Formulation Calculator Molarity Calculator Molecular Weight Calculator Reconstitution Calculator |