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PD 135158

PD 135158

  • CAT Number: I008598
  • CAS Number: 130325-35-8
  • Molecular Formula: C35H44N4O6
  • Molecular Weight: 616.76
  • Purity: ≥95%
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PD 135158 is a Selective cholecystokinin type B (CCKB)/gastrin receptor agonist. In studies, PD- 135158 stimulates lipase release from isolated rat pancreatic acini dose dependently in a biphasic manner, with identical efficacy but lower potency compared to cholecystokinin octapeptide (CCK-8). PD 135158 is classified into Anti-Anxiety Agents, Central Nervous System Agents, Central Nervous System Depressants, Psychotropic Drugs, and Tranquilizing Agents.

Catalog Number I008598
CAS Number 130325-35-8
Molecular Formula

C35H44N4O6

Purity 95%
Target CCK2 Receptors
Solubility Soluble in DMSO
Storage Store at +4C
Reference

</br>1:PD-135158, a CCKB receptor antagonist, microinjected into the nucleus accumbens and the expression of conditioned rewarded behavior. Josselyn SA, Franco VP, Vaccarino FJ.Neurosci Lett. 1996 May 10;209(2):85-8. PMID: 8761988 </br>2:PD 135158, a CCKB/gastrin receptor antagonist, stimulates rat pancreatic enzyme secretion as a CCKA receptor agonist. Höcker M, Hughes J, Fölsch UR, Schmidt WE.Eur J Pharmacol. 1993 Sep 21;242(1):105-8. PMID: 7901038

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