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OT-R antagonist 2

OT-R antagonist 2

  • CAT Number: I003340
  • CAS Number: 364071-16-9
  • Molecular Formula: C28H29N3O4
  • Molecular Weight: 471.557
  • Purity: ≥95%
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<p style=/line-height:25px/>OT-R antagonist 2 is a nonpeptide low molecular weight OT-R antagonist. OT-R antagonist 2 inhibitis IP3-Synthesis, rat OT-R (IC50 = 0.33 μM).<br>IC50 value: 0.33μM<br>Target: oxytocin receptor</p>

Catalog Number I003340
CAS Number 364071-16-9
Molecular Formula

C28H29N3O4

Purity 95%
Target oxytocin receptor
Solubility 10 mM in DMSO
Storage Store at -20C
IC50 0.33μM
IUPAC Name (2S,4E)-N-[(2S)-2-hydroxy-2-phenylethyl]-4-methoxyimino-1-[4-(2-methylphenyl)benzoyl]pyrrolidine-2-carboxamide
InChI InChI=1S/C28H29N3O4/c1-19-8-6-7-11-24(19)20-12-14-22(15-13-20)28(34)31-18-23(30-35-2)16-25(31)27(33)29-17-26(32)21-9-4-3-5-10-21/h3-15,25-26,32H,16-18H2,1-2H3,(H,29,33)/b30-23+/t25-,26+/m0/s1
InChIKey IBXGJPAYWMFXSF-OLFRMSBUSA-N
SMILES CC1=CC=CC=C1C2=CC=C(C=C2)C(=O)N3CC(=NOC)CC3C(=O)NCC(C4=CC=CC=C4)O
Reference

<p style=/line-height:25px/>
<br>[1]. Cirillo R, et al. Pharmacology of (2S,4Z)-N-[(2S)-2-hydroxy-2-phenylethyl]-4-(methoxyimino) -1-[(2/’-methyl[1,1/’-biphenyl]-4-yl)carbonyl]-2-pyrrolidinecarboxamide, a new potent and selective nonpeptide antagonist of the oxytocin receptor. J Pharmacol Exp Ther. 2003 Jul;306(1):253-61.

<br>[2]. William Nadler, et al. Method for preparing pyrrolidine oximes. WO/2005082848/A2.

<br>[3]. Serge Halazy, et al. Pharmaceutically active pyrrolidine derivatives as bax inhibitors.WO/2001074769/A1.

<br>[4]. Serge Halazy, et al. Pharmaceutically active pyrrolidine derivatives as bax inhibitors. WO/2001072705/A1.

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