Orphenadrine citrate

• CAT Number: I003622
• CAS Number: 4682-36-4
• Molecular Formula: C18H23NO.C6H8O7
• Molecular Weight: 461.5
• Purity: ≥95%
• Synonyms: N,N-dimethyl-2-[(2-methylphenyl)-phenylmethoxy]ethanamine;2-hydroxypropane-1,2,3-tricarboxylic acid
• Target: Neuronal Signaling
• Solubility: DMSO 92 mg/mL; Water <1 mg/mL
• Storage: 3 years -20C powder

Orphenadrine citrate (Cat.No:I003622) is a medication primarily used as a muscle relaxant to treat muscle spasms and associated pain. It works by blocking certain nerve impulses that cause muscle contractions. Orphenadrine citrate is also prescribed for the management of Parkinson’s disease and as an adjunct therapy for pain relief.

Reference

[1]. Kornhuber, J., et al., Orphenadrine is an uncompetitive N-methyl-D-aspartate (NMDA) receptor antagonist: binding and patch clamp studies. J Neural Transm Gen Sect, 1995. 102(3): p. 237-46.
[2]. Pubill, D., et al., Assessment of the adrenergic effects of orphenadrine in rat vas deferens. J Pharm Pharmacol, 1999. 51(3): p. 307-12.