MGCD-265 analog

  • CAT Number: I005271
  • CAS Number: 875337-44-3
  • Molecular Formula: C26H20FN5O2S2
  • Molecular Weight: 517.6
  • Purity: ≥95%
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MGCD-265-analog (Cat.No:I005271) (structurally related to MGCD-265) is an orally bioavailable multitargeted tyrosine kinase inhibitor with potential antineoplastic activity with IC50 of 29 nM and 10 nM for c-Met and VEGFR2, respectively.

Catalog Number I005271
CAS Number 875337-44-3
Molecular Formula

C26H20FN5O2S2

Purity 95%
Target Tie-2
Solubility 10 mM in DMSO
Storage 3 years -20C powder
IC50 10 nM (VEGFR2), 29 nM(c-Met) [1]
InChIKey UFICVEHDQUKCEA-UHFFFAOYSA-N
Reference

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