IKK-3 Inhibitor

• CAT Number: I005172
• CAS Number: 862812-98-4
• Molecular Formula: C22H19N3O5S2
• Molecular Weight: 469.5
• Purity: ≥95%
• Target: IκB/IKK
• Solubility: 10 mM in DMSO
• Storage: Store at -20°C
• IC50: 40 nM
• InChI: InChI=1S/C22H19N3O5S2/c1-28-17-8-15-16(9-18(17)29-2)25(13-24-15)22-10-19(20(11-23)31-22)30-12-14-6-4-5-7-21(14)32(3,26)27/h4-10,13H,12H2,1-3H3
• InChIKey: LDTAHRLHGHFHKP-UHFFFAOYSA-N
• SMILES: CS(C1=C(COC2=C(C#N)SC(N3C=NC4=CC(OC)=C(OC)C=C43)=C2)C=CC=C1)(=O)=O

IKK-3 inhibitor (Cat.No:I005172) is a small molecule compound that selectively inhibits the activity of the IKK-ε kinase, also known as IKK-3. This enzyme plays a crucial role in the regulation of immune responses and inflammation. By blocking IKK-3, this inhibitor has potential therapeutic applications in inflammatory diseases and cancer treatment.

Reference

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