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GSK 789472 hydrochloride

GSK 789472 hydrochloride

  • CAT Number: I010857
  • CAS Number: 1257326-24-1
  • Molecular Formula: C15H22ClN3O
  • Molecular Weight: 295.811
  • Purity: ≥95%
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GSK 789472 hydrochloride(CAT: I010857) acts as a selective antagonist of the dopamine D3 receptor and a partial agonist of the dopamine D2 receptor. The compound demonstrates higher potency in antagonizing the D3 receptor (pEC50 < 5.5) compared to its partial agonist activity at the D2 receptor (pEC50 = 8.3). GSK 789472 hydrochloride exhibits selectivity against the dopamine D4 receptor in both agonist and antagonist assays. Importantly, it has the ability to cross the blood-brain barrier, suggesting its potential for central nervous system (CNS) activity.

Catalog Number I010857
CAS Number 1257326-24-1
Molecular Formula

C15H22ClN3O

Purity 95%
Target Dopamine Receptor
Solubility Soluble to 100 mM in water and to 100 mM in DMSO
Storage Desiccate at RT
IUPAC Name 1-phenyl-3-(piperidin-2-ylmethyl)imidazolidin-2-one;hydrochloride
InChI InChI=1S/C15H21N3O.ClH/c19-15-17(12-13-6-4-5-9-16-13)10-11-18(15)14-7-2-1-3-8-14;/h1-3,7-8,13,16H,4-6,9-12H2;1H
InChIKey BYJUVPWUMBVSTK-UHFFFAOYSA-N
SMILES C1CCNC(C1)CN2CCN(C2=O)C3=CC=CC=C3.Cl

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