Gabapentin

• CAT Number: I004258
• CAS Number: 60142-96-3
• Molecular Formula: C9H17NO2
• Molecular Weight: 171.2
• Purity: ≥95%
• Target: GABA Receptor
• Solubility: H2O: 34 mg/mL, DMSO: ＜1 mg/mL
• Storage: 3 years -20C powder
• IC50: 140 nM (α2δ subunit of calcium channel) [1]
• IUPAC Name: 2-[1-(aminomethyl)cyclohexyl]acetic acid
• InChI: InChI=1S/C9H17NO2/c10-7-9(6-8(11)12)4-2-1-3-5-9/h1-7,10H2,(H,11,12)
• InChIKey: UGJMXCAKCUNAIE-UHFFFAOYSA-N

Gabapentin (CAT: I004258) is a medication used primarily to treat epilepsy and neuropathic pain. It belongs to the class of anticonvulsant drugs and works by affecting the chemicals and nerves in the body that are involved in seizures and pain signals. Gabapentin is thought to modulate the activity of certain neurotransmitters, such as gamma-aminobutyric acid (GABA), in the brain, which helps to reduce abnormal electrical activity and alleviate pain. In addition to its approved uses, gabapentin may also be prescribed off-label for other conditions, including anxiety disorders and restless legs syndrome.

Reference

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