CONTACT US
Home > Inhibitors/Agonists> > DR 4485 hydrochloride
DR 4485 hydrochloride

DR 4485 hydrochloride

  • CAT Number: I011074
  • CAS Number: 402942-53-4
  • Molecular Formula: C26H29Cl3N2O
  • Molecular Weight: 491.881
  • Purity: ≥95%
Inquiry Now

High affinity and selective 5-HT<sub>7</sub> antagonist (pK<sub>i</sub> = 8.14). Exhibits selectivity for 5-HT<sub>7</sub> over other 5-HT receptors. Inhibits 5-HT-induced cAMP accumulation in HEK-293 cells expressing the 5-HT<sub>7</sub> receptor. Orally bioavailable.

Catalog Number I011074
CAS Number 402942-53-4
Synonyms

6-Chloro-2a-[4-[4-(4-chlorophenyl)-3,6-dihydro-1(2H)-pyridinyl]butyl]-2a,3,4,5-tetrahydrobenz[cd]indol-2(1H)-one hydrochloride

Molecular Formula

C26H29Cl3N2O

Purity 95%
Target 5-HT Receptor
Solubility Soluble to 100 mM in DMSO
Storage Desiccate at RT
IUPAC Name 6-chloro-2a-[4-[4-(4-chlorophenyl)-3,6-dihydro-2H-pyridin-1-yl]butyl]-1,3,4,5-tetrahydrobenzo[cd]indol-2-one;hydrochloride
InChI InChI=1S/C26H28Cl2N2O.ClH/c27-20-7-5-18(6-8-20)19-11-16-30(17-12-19)15-2-1-13-26-14-3-4-21-22(28)9-10-23(24(21)26)29-25(26)31;/h5-11H,1-4,12-17H2,(H,29,31);1H
InChIKey QAERYGXKDZHTFR-UHFFFAOYSA-N
SMILES C1CC2=C(C=CC3=C2C(C1)(C(=O)N3)CCCCN4CCC(=CC4)C5=CC=C(C=C5)Cl)Cl.Cl

Request a Quote

Contact Us at MuseChem

We are committed to providing you with reliable, cost-effective solutions for your chemical needs, while ensuring your safety and comfort. Our team of experts is always available to answer your questions and help you navigate the complexities of the chemical industry.

Whether you're looking for a specific product or need help with a custom synthesis project, we're here to help you discover a new world of chemical possibilities. Contact us today to learn more about how we can assist you with all of your chemical needs.

Our goal is to make the process of ordering chemicals as seamless and hassle-free as possible. Let us know how we can assist you, and we'll get back to you as soon as possible. We look forward to hearing from you!