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Cgp 11130

Cgp 11130

  • CAT Number: I005966
  • CAS Number: 52237-19-1
  • Molecular Formula: C10H12FNO2
  • Molecular Weight: 197.209
  • Purity: 98%
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<span style="color:#000000;"><span style="font-size:12px;"><span style="font-family:arial,helvetica,sans-serif;">Cgp 11130 (CAS&nbsp;52237-19-1) is a bio-active chemical. It&nbsp;is a GABAB receptor agonist which was never marketed. It is selective for the GABAB receptor over the GABAA receptor (IC50 = 1.70 &mu;M and &gt; 100 &mu;M, respectively). The drug is a GABA analogue and is closely related to baclofen (&beta;-(4-chlorophenyl)-GABA), tolibut (&beta;-(4-methylphenyl)-GABA), and phenibut (&beta;-phenyl-GABA). It is less potent as a GABAB receptor agonist than baclofen but more potent than phenibut.</span></span></span></p>
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Catalog Number I005966
CAS Number 52237-19-1
Molecular Formula

C10H12FNO2

Purity 98
Solubility Soluble in DMSO, not in water
Storage 0 - 4°C for short term ,or -20 °C for long term
Related CAS 1858241-03-8(hydrochloride)
IUPAC Name 4-amino-3-(4-fluorophenyl)butanoic acid
InChI InChI=1S/C10H12FNO2/c11-9-3-1-7(2-4-9)8(6-12)5-10(13)14/h1-4,8H,5-6,12H2,(H,13,14)
InChIKey QWHXHLDNSXLAPX-UHFFFAOYSA-N
SMILES C1=CC(=CC=C1C(CC(=O)O)CN)F
Reference

<span style="color:#000000;"><span style="font-size:12px;"><span style="font-family:arial,helvetica,sans-serif;">1.Spahn, Hildegard, Dorit Krau&beta;, and Ernst Mutschler. &quot;Enantiospecific high-performance liquid chromatographic (HPLC) determination of baclofen and its fluoro analogue in biological material.&quot;&nbsp;<i style="font-family: Arial, sans-serif; font-size: 13px;">Pharmaceutical research</i>&nbsp;5.2 (1988): 107-112.</span></span></span>

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