Busulfan

• CAT Number: A000926
• CAS Number: 55-98-1
• Molecular Formula: C6H14O6S2
• Molecular Weight: 246.3
• Purity: ≥95%
• Target: DNA Alkylating
• Solubility: >12.3mg/mL in DMSO
• Storage: -20°C
• InChI: 1S/C6H14O6S2/c1-13(7,8)11-5-3-4-6-12-14(2,9)10/h3-6H2,1-2H3
• InChIKey: COVZYZSDYWQREU-UHFFFAOYSA-N
• SMILES: CS(=O)(=O)OCCCCOS(=O)(=O)C

Busulfan (Myleran, GlaxoSmithKline, Busulfex IV, Otsuka America Pharmaceutical, Inc.) is a cancer drug, in use since 1959. Busulfan is a cell cycle non-specific alkylating antineoplastic agent, in the class of alkyl sulfonates. Its chemical designation is 1,4-butanediol dimethanesulfonate.

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