ARP100

• CAT Number: I002786
• CAS Number: 704888-90-4
• Molecular Formula: C17H20N2O5S
• Molecular Weight: 364.416
• Purity: ≥95%
• Target: MMP
• Solubility: Soluble in DMSO
• Storage: 0 - 4°Cfor short term (days to weeks), or -20 °C for long term (months).
• IUPAC Name: N-hydroxy-2-[(4-phenylphenyl)sulfonyl-propan-2-yloxyamino]acetamide
• InChI: InChI=1S/C17H20N2O5S/c1-13(2)24-19(12-17(20)18-21)25(22,23)16-10-8-15(9-11-16)14-6-4-3-5-7-14/h3-11,13,21H,12H2,1-2H3,(H,18,20)
• InChIKey: PHGLPDURIUEELR-UHFFFAOYSA-N
• SMILES: CC(C)ON(CC(=O)NO)S(=O)(=O)C1=CC=C(C=C1)C2=CC=CC=C2

ARP100 (CAT: I002786) is a specific inhibitor targeting matrix metalloproteinase-2 (MMP-2), an enzyme involved in extracellular matrix remodeling. By selectively inhibiting MMP-2, ARP100 can potentially impact various processes such as tissue remodeling, wound healing, and angiogenesis. This selective inhibition could have applications in controlling pathological conditions where MMP-2 activity plays a significant role, such as cancer metastasis and tissue fibrosis.

Reference

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