Valsartan

• CAT Number: A000712
• CAS Number: 137862-53-4
• Molecular Formula: C₂₄H₂₉N₅O₃
• Molecular Weight: 435.52
• Purity: ≥95%
• Synonyms: 137862-53-4; Diovan; Provas; Tareg; L-Valsartan
• Target: Angiotensin Receptor
• Solubility: >19.7mg/mL in DMSO
• Storage: -20°C
• IUPAC Name: (2S)-3-methyl-2-[pentanoyl-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]amino]butanoic acid
• InChI: InChI=1S/C24H29N5O3/c1-4-5-10-21(30)29(22(16(2)3)24(31)32)15-17-11-13-18(14-12-17)19-8-6-7-9-20(19)23-25-27-28-26-23/h6-9,11-14,16,22H,4-5,10,15H2,1-3H3,(H,31,32)(H,25,26,27,28)/t22-/m0/s1
• InChIKey: ACWBQPMHZXGDFX-QFIPXVFZSA-N
• SMILES: CCCCC(=O)N(CC1=CC=C(C=C1)C2=CC=CC=C2C3=NNN=N3)[C@@H](C(C)C)C(=O)O

Valsartan（Cat No.:A000712）is an angiotensin II receptor blocker (ARB) with the chemical formula C24H29N5O3, used primarily to treat high blood pressure, heart failure, and to improve survival after heart attacks. By selectively blocking the angiotensin II type 1 (AT1) receptor, it prevents vasoconstriction and aldosterone secretion, thereby lowering blood pressure and reducing cardiac workload. Valsartan is administered orally and is well-absorbed, though bioavailability is moderate. It is often prescribed alone or in combination with other antihypertensives. Valsartan is generally well tolerated and plays a key role in cardiovascular disease management.

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