For research use only. Not for therapeutic Use.
UNC2541（Cat No.:I019010）is a selective small-molecule inhibitor of the bromodomain and extra-terminal (BET) family protein BRD4, a key regulator of gene transcription linked to cancer progression and inflammatory signaling. By binding to the acetyl-lysine recognition pocket of BRD4, UNC2541 disrupts transcriptional programs controlling cell growth and survival. This compound is widely used in oncology and epigenetics research to study BET-dependent signaling, transcriptional regulation, and potential therapeutic strategies. UNC2541 provides researchers with a precise tool to investigate BRD4 biology and develop novel approaches for cancer and inflammation treatment.
| CAS Number | 1612782-86-1 |
| Synonyms | (7S)-7-amino-N-[(4-fluorophenyl)methyl]-8-oxo-2,9,16,18,21-pentazabicyclo[15.3.1]henicosa-1(21),17,19-triene-20-carboxamide |
| Molecular Formula | C24H34FN7O2 |
| Purity | ≥95% |
| IUPAC Name | (7S)-7-amino-N-[(4-fluorophenyl)methyl]-8-oxo-2,9,16,18,21-pentazabicyclo[15.3.1]henicosa-1(21),17,19-triene-20-carboxamide |
| InChI | InChI=1S/C24H34FN7O2/c25-18-10-8-17(9-11-18)15-30-22(33)19-16-31-24-29-14-5-2-1-4-13-28-23(34)20(26)7-3-6-12-27-21(19)32-24/h8-11,16,20H,1-7,12-15,26H2,(H,28,34)(H,30,33)(H2,27,29,31,32)/t20-/m0/s1 |
| InChIKey | ONIHBIZGUJZDHG-FQEVSTJZSA-N |
| SMILES | C1CCCNC2=NC=C(C(=N2)NCCCC[C@@H](C(=O)NCC1)N)C(=O)NCC3=CC=C(C=C3)F |
| Chemistry Calculators | Dilution Calculator In vivo Formulation Calculator Molarity Calculator Molecular Weight Calculator Reconstitution Calculator |
