Teneligliptin hydrobromide hydrate

  • CAT Number: I018947
  • CAS Number: 1572583-29-9
  • Molecular Formula: C₂₂H₃₀N₆OS
  • Molecular Weight: 426.58
  • Purity: ≥95%
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Tiniletine hydrobromide hydrate (Cat No.:I018947) is a potent chemotypic prolylthiazoline DPP-4 inhibitor that competitively inhibits human plasma, rat plasma, and human recombinant DPP-4 in vitro with an IC50 of approximately 1 nM.

Catalog Number I018947
CAS Number 1572583-29-9
Molecular Formula

C₂₂H₃₀N₆OS

Purity 95%
Reference

[1]. Fukuda-Tsuru S, et al. A novel, potent, and long-lasting dipeptidyl peptidase-4 inhibitor, teneligliptin, improves postprandial hyperglycemia and dyslipidemia after single and repeated administrations. Eur J Pharmacol. 2012 Dec 5;696(1-3):194-202.

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