Pipendoxifene

• CAT Number: R045574
• CAS Number: 198480-55-6
• Molecular Formula: C29H32N2O3
• Molecular Weight: 456.58
• Purity: ≥95%
• Storage: Store at RT
• IUPAC Name: 2-(4-hydroxyphenyl)-3-methyl-1-[[4-(2-piperidin-1-ylethoxy)phenyl]methyl]indol-5-ol
• InChI: InChI=1S/C29H32N2O3/c1-21-27-19-25(33)11-14-28(27)31(29(21)23-7-9-24(32)10-8-23)20-22-5-12-26(13-6-22)34-18-17-30-15-3-2-4-16-30/h5-14,19,32-33H,2-4,15-18,20H2,1H3
• InChIKey: JICOGKJOQXTAIP-UHFFFAOYSA-N
• SMILES: CC1=C(N(C2=C1C=C(C=C2)O)CC3=CC=C(C=C3)OCCN4CCCCC4)C5=CC=C(C=C5)O

Pipendoxifene（Cat No.:R045574）, is a synthetic selective estrogen receptor modulator (SERM) that has been studied for its potential in hormone-related therapies, particularly in breast cancer treatment and osteoporosis management. As a SERM, pipendoxifene interacts with estrogen receptors in a tissue-specific manner, acting as an agonist or antagonist depending on the target tissue. This property allows it to provide estrogen-like effects in bone tissue, beneficial for preventing osteoporosis, while acting as an antagonist in breast tissue, potentially reducing the risk of estrogen-driven breast cancer.

Reference

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