For research use only. Not for therapeutic Use.
MRS2500 tetraammonium(Cat No.:R014564)is a potent, selective antagonist of the purinergic P2Y1 receptor, a G-protein–coupled receptor activated by ADP and involved in platelet aggregation and thrombosis. By blocking P2Y1 signaling, MRS2500 effectively inhibits platelet activation and aggregation, making it a valuable research tool in cardiovascular and hematology studies. It is widely used to explore platelet function, purinergic signaling pathways, and potential therapeutic strategies for antithrombotic interventions. Its high affinity and selectivity for P2Y1 provide researchers with precise control in studying platelet-driven vascular and thrombotic disorders.
CAS Number | 630103-23-0 |
Synonyms | diamino [(1R,2S,4S,5S)-2-diaminooxyphosphoryloxy-4-[2-iodo-6-(methylamino)purin-9-yl]-1-bicyclo[3.1.0]hexanyl]methyl phosphate |
Molecular Formula | C13H30IN9O8P2 |
Purity | ≥95% |
IUPAC Name | azane;[(1R,2S,4S,5S)-4-[2-iodo-6-(methylamino)purin-9-yl]-2-phosphonooxy-1-bicyclo[3.1.0]hexanyl]methyl dihydrogen phosphate |
InChI | InChI=1S/C13H18IN5O8P2.4H3N/c1-15-10-9-11(18-12(14)17-10)19(5-16-9)7-2-8(27-29(23,24)25)13(3-6(7)13)4-26-28(20,21)22;;;;/h5-8H,2-4H2,1H3,(H,15,17,18)(H2,20,21,22)(H2,23,24,25);4*1H3/t6-,7+,8+,13+;;;;/m1..../s1 |
InChIKey | FVTFHHDVLNQSME-AVAGOIHISA-N |
SMILES | CNC1=C2C(=NC(=N1)I)N(C=N2)[C@H]3C[C@@H]([C@]4([C@@H]3C4)COP(=O)(O)O)OP(=O)(O)O.N.N.N.N |
Chemistry Calculators | Dilution Calculator In vivo Formulation Calculator Molarity Calculator Molecular Weight Calculator Reconstitution Calculator |