For research use only. Not for therapeutic Use.
Morphiceptin（Cat No.:I044312）is a synthetic tetrapeptide with the sequence Tyr-Pro-Phe-Pro, known for its potent and selective agonist activity at the mu-opioid receptor (MOR). It mimics the action of endogenous opioid peptides, producing analgesic effects by inhibiting pain signaling in the central nervous system. Due to its high receptor selectivity, morphiceptin is widely used in pharmacological studies to investigate opioid receptor function, pain modulation, and the development of safer opioid-based therapeutics. Its small size and defined activity make it a valuable tool in neuropharmacology and analgesic drug discovery research.
| CAS Number | 74135-04-9 |
| Synonyms | (2S)-1-[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]-N-[(2S)-1-[(2S)-2-carbamoylpyrrolidin-1-yl]-1-oxo-3-phenylpropan-2-yl]pyrrolidine-2-carboxamide |
| Molecular Formula | C28H35N5O5 |
| Purity | ≥95% |
| IUPAC Name | (2S)-1-[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]-N-[(2S)-1-[(2S)-2-carbamoylpyrrolidin-1-yl]-1-oxo-3-phenylpropan-2-yl]pyrrolidine-2-carboxamide |
| InChI | InChI=1S/C28H35N5O5/c29-21(16-19-10-12-20(34)13-11-19)27(37)33-15-5-9-24(33)26(36)31-22(17-18-6-2-1-3-7-18)28(38)32-14-4-8-23(32)25(30)35/h1-3,6-7,10-13,21-24,34H,4-5,8-9,14-17,29H2,(H2,30,35)(H,31,36)/t21-,22-,23-,24-/m0/s1 |
| InChIKey | LSQXZIUREIDSHZ-ZJZGAYNASA-N |
| SMILES | C1C[C@H](N(C1)C(=O)[C@H](CC2=CC=C(C=C2)O)N)C(=O)N[C@@H](CC3=CC=CC=C3)C(=O)N4CCC[C@H]4C(=O)N |
| Chemistry Calculators | Dilution Calculator In vivo Formulation Calculator Molarity Calculator Molecular Weight Calculator Reconstitution Calculator |
