For research use only. Not for therapeutic Use.
L002（Cat No.:R030153）is a potent small-molecule inhibitor of p300 histone acetyltransferase (HAT), an epigenetic regulator that acetylates histones and transcription factors to control gene expression. By blocking p300 activity, L002 disrupts acetylation-dependent signaling pathways, leading to altered transcriptional regulation of genes involved in cancer, inflammation, and cell growth. It has demonstrated antiproliferative effects in tumor models and is widely used to study epigenetic control mechanisms. L002 serves as a valuable pharmacological tool for exploring therapeutic strategies targeting histone acetylation in oncology and inflammatory disease research.
| CAS Number | 321695-57-2 |
| Synonyms | [(3,5-dimethyl-4-oxocyclohexa-2,5-dien-1-ylidene)amino] 4-methoxybenzenesulfonate |
| Molecular Formula | C15H15NO5S |
| Purity | ≥95% |
| IUPAC Name | [(3,5-dimethyl-4-oxocyclohexa-2,5-dien-1-ylidene)amino] 4-methoxybenzenesulfonate |
| InChI | InChI=1S/C15H15NO5S/c1-10-8-12(9-11(2)15(10)17)16-21-22(18,19)14-6-4-13(20-3)5-7-14/h4-9H,1-3H3 |
| InChIKey | VEWFTYOFWIXCIO-UHFFFAOYSA-N |
| SMILES | CC1=CC(=NOS(=O)(=O)C2=CC=C(C=C2)OC)C=C(C1=O)C |
| Chemistry Calculators | Dilution Calculator In vivo Formulation Calculator Molarity Calculator Molecular Weight Calculator Reconstitution Calculator |
