For research use only. Not for therapeutic Use.
EP2 receptor antagonist-1（Cat No.:I045076）is a selective inhibitor targeting the prostaglandin E2 receptor subtype EP2, which plays a key role in inflammation, pain, tumor progression, and neurodegeneration. By blocking EP2 receptor signaling, this compound reduces cAMP-mediated pathways involved in pro-inflammatory cytokine release and immune cell activation. EP2 receptor antagonist-1 has shown potential in preclinical models for treating conditions such as Alzheimer’s disease, osteoarthritis, and certain cancers. Its high selectivity and favorable pharmacokinetics make it a promising candidate for modulating prostaglandin-driven pathological processes with minimized off-target effects.
| CAS Number | 848920-08-1 |
| Synonyms | oxolan-2-ylmethyl 2-amino-1-(2,3-dihydro-1,4-benzodioxin-6-yl)pyrrolo[3,2-b]quinoxaline-3-carboxylate |
| Molecular Formula | C24H22N4O5 |
| Purity | ≥95% |
| IUPAC Name | oxolan-2-ylmethyl 2-amino-1-(2,3-dihydro-1,4-benzodioxin-6-yl)pyrrolo[3,2-b]quinoxaline-3-carboxylate |
| InChI | InChI=1S/C24H22N4O5/c25-22-20(24(29)33-13-15-4-3-9-30-15)21-23(27-17-6-2-1-5-16(17)26-21)28(22)14-7-8-18-19(12-14)32-11-10-31-18/h1-2,5-8,12,15H,3-4,9-11,13,25H2 |
| InChIKey | OHXALKVNKANGKL-UHFFFAOYSA-N |
| SMILES | C1CC(OC1)COC(=O)C2=C(N(C3=NC4=CC=CC=C4N=C23)C5=CC6=C(C=C5)OCCO6)N |
| Chemistry Calculators | Dilution Calculator In vivo Formulation Calculator Molarity Calculator Molecular Weight Calculator Reconstitution Calculator |
