Centchroman

• CAT Number: R058485
• CAS Number: 31477-60-8
• Molecular Formula: C30H35NO3
• Molecular Weight: 457.614
• Purity: ≥95%
• Synonyms: rel-1-[2-[4-[(3R,4R)-3,4-dihydro-7-methoxy-2,2-dimethyl-3-phenyl-2H-1-benzopyran-4-yl]phenoxy]ethyl]pyrrolidine; 1-[2-[p-(trans-7-Methoxy-2,2-dimethyl-3-phenyl-4-chromanyl)phenoxy]ethyl]pyrrolidine; 3,4-trans-2,2-Dimethyl-3-phenyl-4-[p-(β-pyrrolidi
• Target: Estrogen/progestogen Receptor
• Solubility: Soluble in DMSO
• Storage: Store at -20°C
• IUPAC Name: 1-[2-[4-[(3S,4S)-7-methoxy-2,2-dimethyl-3-phenyl-3,4-dihydrochromen-4-yl]phenoxy]ethyl]pyrrolidine
• InChI: InChI=1S/C30H35NO3/c1-30(2)29(23-9-5-4-6-10-23)28(26-16-15-25(32-3)21-27(26)34-30)22-11-13-24(14-12-22)33-20-19-31-17-7-8-18-31/h4-6,9-16,21,28-29H,7-8,17-20H2,1-3H3/t28-,29+/m0/s1
• InChIKey: XZEUAXYWNKYKPL-URLMMPGGSA-N
• SMILES: CC1(C(C(C2=C(O1)C=C(C=C2)OC)C3=CC=C(C=C3)OCCN4CCCC4)C5=CC=CC=C5)C

Centchroman, also known as Ormeloxifene, is a non-steroidal oral contraceptive used primarily in India. It functions uniquely by modulating the estrogen receptors, rather than the traditional hormonal suppression of ovulation. Centchroman serves as a selective estrogen receptor modulator (SERM), providing a safer profile with fewer hormonal side effects compared to conventional birth control pills. It also exhibits therapeutic benefits in the treatment of dysfunctional uterine bleeding and as a potential agent in breast cancer prevention.