For research use only. Not for therapeutic Use.
BRD0209（Cat No.:I023657）is a selective small-molecule inhibitor targeting bromodomain-containing proteins, particularly within the BET (bromodomain and extra-terminal) family. By disrupting the interaction between BET proteins and acetylated histones, BRD0209 modulates transcription of key oncogenes such as MYC, thereby exhibiting antiproliferative and pro-apoptotic effects in cancer models. It is used extensively in epigenetics research to investigate chromatin remodeling, transcriptional regulation, and BET-dependent gene expression. BRD0209 serves as a valuable tool for studying BET protein functions and exploring therapeutic strategies in oncology, inflammation, and other transcriptionally driven diseases.
| CAS Number | 1597439-87-6 |
| Synonyms | (4S)-3-cyclopropyl-4,7,7-trimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one |
| Molecular Formula | C22H25N3O |
| Purity | ≥95% |
| IUPAC Name | (4S)-3-cyclopropyl-4,7,7-trimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one |
| InChI | InChI=1S/C22H25N3O/c1-21(2)11-15-17(16(26)12-21)22(3,14-7-5-4-6-8-14)18-19(13-9-10-13)24-25-20(18)23-15/h4-8,13H,9-12H2,1-3H3,(H2,23,24,25)/t22-/m1/s1 |
| InChIKey | YKPIWOGXCSQLFH-JOCHJYFZSA-N |
| SMILES | C[C@]1(C2=C(CC(CC2=O)(C)C)NC3=NNC(=C31)C4CC4)C5=CC=CC=C5 |
| Chemistry Calculators | Dilution Calculator In vivo Formulation Calculator Molarity Calculator Molecular Weight Calculator Reconstitution Calculator |
