Apatinib-d8 Hydrochloride

• CAT Number: C000565
• CAS Number: 2468771-44-8
• Molecular Formula: C₂₄H₁₅D₈N₅O • HCl
• Molecular Weight: 441.98
• Purity: ≥95%
• Synonyms: N-[4-(1-Cyanocyclopentyl-d8)phenyl]-2-[(4-pyridinylmethyl)amino]-3-pyridinecarboxamide; YN968D1-d8 Hydrochloride
• Solubility: DMSO (Slightly), Methanol (Slightly)
• Storage: 4°C

Apatinib-d8 Hydrochloride (CAT: C000565) is a deuterated derivative of Apatinib Hydrochloride, a tyrosine kinase inhibitor used in pharmaceutical research. It functions by selectively targeting and inhibiting the vascular endothelial growth factor receptor-2 (VEGFR-2), a key player in angiogenesis. In the pharmaceutical field, Apatinib-d8 Hydrochloride is a valuable tool compound for studying anti-angiogenic mechanisms and drug interactions. Its stable isotopic labeling with deuterium can aid in drug metabolism and pharmacokinetic studies, making it an asset in drug development research.

Reference

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