Amidopyrine

• CAT Number: A000220
• CAS Number: 58-15-1
• Molecular Formula: C13H17N3O
• Molecular Weight: 231.29
• Purity: ≥95%
• Storage: -20°C
• InChI: 1S/C13H17N3O/c1-10-12(14(2)3)13(17)16(15(10)4)11-8-6-5-7-9-11/h5-9H,1-4H3
• InChIKey: RMMXTBMQSGEXHJ-UHFFFAOYSA-N
• SMILES: CC1=C(C(=O)N(N1C)C2=CC=CC=C2)N(C)C

Aminophenazone, also known as aminopyrine, is a non-steroidal anti-inflammatory drugs used to treat pain and inflammation.

Reference

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models of amidopyrine and its metabolites in complexes with rabbit cytochrome
P450 2B4 reveal a structural mechanism of sequential N-dealkylation.
Biochemistry. 2011 Mar 29;50(12):2123-34. doi: 10.1021/bi101797v. Epub 2011 Mar
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2: Petrenko AIu, Povolotskaia VA, Rosliakov AD, Libina VV, Chaĭka LA.
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5: Noskov SM. [Megaloblastic pancytopenia in a female patient with rheumatoid
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6: Moroz BT, Ignatov IuD, Kalinin VI. [Thresholds of the electrical excitability
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7: Adrianov NV, Dovgiĭ AI, Khaĭlov PM. [The effect of phenobarbital and
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8: Savchenko MV, Ivanova LA. [Use of amidopyrine for assessing thiourea exposure
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9: Bai T, Jia JH. [Application of the derivative linear regression method of
multiwavelength data to the simultaneous determination of amidopyrine and
caffeine in compound amidopyrine and caffeine tablets]. Yao Xue Xue Bao.
1988;23(8):616-22. Chinese. PubMed PMID: 3254043.

10: Tarakhovskiĭ ML, Zaĭtseva NE, Mozalevskiĭ AF. [Individual characteristics and
effects of spasmolytics in relation to the oxidation phenotype of the marker
preparation amidopyrine in children with digestive and respiratory diseases].
Pediatriia. 1988;(4):43-7. Russian. PubMed PMID: 3205647.